Biochemistry

DPP-4

Dipeptidyl peptidase-4 — a protease that rapidly degrades native GLP-1 and GIP.

Definition

DPP-4 cleaves peptides at the N-terminal second position after proline or alanine. Native GLP-1 has a half-life of ~2 minutes due to DPP-4. GLP-1 analogs (semaglutide, liraglutide) are engineered to resist DPP-4 cleavage.

Related terms

Back to the full peptide glossary.