Pharmacology
Glucagon Receptor
GPCR that regulates hepatic glucose production; co-activated by triple agonists like retatrutide.
Definition
The glucagon receptor (GCGR) opposes insulin action by promoting hepatic glucose production and lipolysis. Triple agonists add glucagon receptor activation to increase energy expenditure and accelerate hepatic fat oxidation.
Related terms
Compounds that reference Glucagon Receptor
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