Biochemistry

Protease

An enzyme that cleaves peptide bonds, breaking peptides into smaller fragments.

Definition

Proteases (endopeptidases, exopeptidases) include DPP-4, neprilysin, trypsin, and chymotrypsin. Peptide drug design frequently targets resistance to specific proteases — e.g., semaglutide's acyl chain shields it from DPP-4.

Related terms

Back to the full peptide glossary.